| IUPAC name | 1-butyl-N-(2,6-dimethylphenyl)piperidine-2-carboxamide;hydrate;hydrochloride |
| inchi | InChI=1S/C18H28N2O.ClH.H2O/c1-4-5-12-20-13-7-6-11-16(20)18(21)19-17-14(2)9-8-10-15(17)3;;/h8-10,16H,4-7,11-13H2,1-3H3,(H,19,21);1H;1H2 |
| inchi key | HUCIWBPMHXGLFM-UHFFFAOYSA-N |
| molecular formula | C18H31ClN2O2 |
| synonyms | 73360-54-0Bupivacaine hydrochloride monohydrateSensorcaineBupivacaine hydrochloride hydrateWIN-11318 |
| Compound Description | Bupivacaine hydrochloride hydrate is a racemate composed of equimolar amounts of dextrobupivacaine hydrochloride hydrate and levobupivacaine hydrochloride hydrate. A piperidinecarboxamide-based local anaesthetic, it has a slow onset and long duration of action. It has a role as a local anaesthetic, an adrenergic antagonist, an amphiphile, an EC 3.1.1.8 inhibitor and an EC 3.6.3.8 -transporting ATPase) inhibitor. It contains a bupivacaine hydrochloride , a levobupivacaine hydrochloride hydrate and a dextrobupivacaine hydrochloride hydrate.Bupivacaine Hydrochloride is a long-acting, amide-type local anesthetic. Bupivicaine reversibly binds to specific sodium ion channels in the neuronal membrane, resulting in a decrease in the voltage-dependent membrane permeability to sodium ions and membrane stabilization; inhibition of depolarization and nerve impulse conduction; and a reversible loss of sensation.A widely used local anesthetic agent. |
